SCHEMBL3374792

SCHEMBL3374792

O=C(N[C@H]1CCC[C@@](O)(C#Cc2cccc(Cl)c2)C1)Oc1ccc(Cl)o1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 15/20 0.46
EPHX2 P34913 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3373020 1.00 GRM5 (0.46) GRM5EPHX2L3MBTL1NPC1RAB9A
SCHEMBL3374718 0.87 GRM5 (0.46) GRM5EPHX2L3MBTL1NPC1RAB9A
SCHEMBL3374694 0.87 GRM5 (0.46) GRM5EPHX2L3MBTL1NPC1RAB9A
SCHEMBL3376495 0.86 GRM5 (0.43) GRM5NPC1RAB9A
SCHEMBL3376064 0.86 GRM5 (0.44) GRM5EPHX2L3MBTL1NPC1RAB9A
SCHEMBL3374797 0.86 GRM5 (0.44) GRM5EPHX2L3MBTL1NPC1RAB9A
SCHEMBL991006 0.84 GRM5 (0.46) GRM5L3MBTL1NPC1RAB9A
SCHEMBL992693 0.84 GRM5 (0.46) GRM5L3MBTL1NPC1RAB9A
SCHEMBL3379028 0.84 GRM5 (0.46) GRM5
SCHEMBL3375912 0.84 GRM5 (0.46) GRM5EPHX2L3MBTL1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877365-B1 ACETYLENE DERIVATIVES NOVARTIS AG (CH) 2010-11-10 EP claimed