SCHEMBL3375341

SCHEMBL3375341

Cc1cc(SC/C=C(\C#CCO)c2ccc(Br)cc2)ccc1O

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 4/20 0.44
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
STAT6 P42226 1/20 0.35
HSP90AA1 P07900 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3372729 0.87 PPARD (0.34) PPARDALDH1A1HSP90AA1
SCHEMBL3375669 0.84 PPARD (0.44) PPARDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL3026125 0.81 PPARD (0.71) PPARD
SCHEMBL3021922 0.79 PPARD (0.49) PPARDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL3021925 0.79 PPARD (0.49) PPARDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL3372723 0.75 PPARD (0.36) PPARDALDH1A1
SCHEMBL3375667 0.72 PPARD (0.46) PPARDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL3266067 0.71 PPARD (0.55) PPARDALDH1A1
SCHEMBL3021862 0.70 PPARD (0.56) PPARD
SCHEMBL3033687 0.70 PPARD (0.56) PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745002-B1 NOVEL COMPOUNDS, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS LLC (US) 2010-11-03 EP claimed
EP-1745002-B1 NOVEL COMPOUNDS, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS LLC (US) 2010-11-03 EP disclosed