SCHEMBL3376814

SCHEMBL3376814

CCOC(=O)C1(CBr)CCC2(CC1)OCCO2

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP2C9 P11712 1/20 0.40
POLB P06746 2/20 0.36
KMT2A Q03164 3/20 0.35
TRPA1 O75762 1/20 0.33
MAPK1 P28482 3/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ATM Q13315 1/20 0.33
LMNA P02545 3/20 0.32
HSD17B10 Q99714 1/20 0.32
MEN1 O00255 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14212551 0.87 ALDH1A1 (0.41) ALDH1A1CYP3A4CYP2C19CYP2C9POLB
SCHEMBL9149710 0.86 ALDH1A1 (0.43) ALDH1A1POLBKMT2ATRPA1MAPK1
SCHEMBL11920271 0.85 ALDH1A1 (0.40) ALDH1A1CYP3A4CYP2C19CYP2C9POLB
SCHEMBL16897503 0.84 ALDH1A1 (0.40) ALDH1A1CYP3A4CYP2C19CYP2C9POLB
SCHEMBL12346121 0.84 ALDH1A1 (0.40) ALDH1A1CYP3A4CYP2C19CYP2C9POLB
SCHEMBL17682272 0.83 ALDH1A1 (0.39) ALDH1A1CYP3A4CYP2C19CYP2C9POLB
SCHEMBL7308023 0.81 TSHR (0.41) ALDH1A1CYP3A4CYP2C19POLBKMT2A
SCHEMBL12161 0.81 ALDH1A1 (0.38) ALDH1A1CYP3A4CYP2C19CYP2C9POLB
SCHEMBL25986067 0.81 ALDH1A1 (0.38) ALDH1A1CYP3A4CYP2C19CYP2C9POLB
SCHEMBL10263 0.80 ALDH1A1 (0.38) ALDH1A1CYP3A4CYP2C19CYP2C9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046388-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUINOLIN-2-ONES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed
US-6503910-B1 Metalloproteinase inhibitors; antimetastasis agents; arthritis, neurodegenerative disorder treatment DARWIN DISCOVERY LTD. (GB) 2003-01-07 US disclosed
EP-1177183-A1 HYDROXAMIC AND CARBOXYLIC ACID DERIVATIVES Darwin Discovery Limited (GB) 2002-02-06 EP disclosed
WO-2000069839-A1 HYDROXAMIC AND CARBOXYLIC ACID DERIVATIVES DARWIN DISCOVERY LIMITED (GB) 2000-11-23 WO disclosed