SCHEMBL3376816

SCHEMBL3376816

COc1ccc2ncc(F)c(C(O)C(O)([C@H]3CC[C@H](NC/C=C/c4cccc(F)c4)CC3)[C@@](O)([C@H]3CC[C@H](NC/C=C/c4cc(F)ccc4F)CC3)[C@H](O)c3c(F)cnc4ccc(OC)nc34)c2n1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.40
SLC2A1 P11166 2/20 0.39
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3374575 0.83 KCNH2 (0.43) KCNH2SLC2A1
SCHEMBL3374578 0.83 KCNH2 (0.43) KCNH2SLC2A1
SCHEMBL3374273 0.83 KCNH2 (0.43) KCNH2SLC2A1
SCHEMBL3374571 0.83 KCNH2 (0.43) KCNH2SLC2A1
SCHEMBL3375784 0.81 KCNH2 (0.44) KCNH2SLC2A1
SCHEMBL3373002 0.81 KCNH2 (0.44) KCNH2SLC2A1
SCHEMBL3373006 0.81 KCNH2 (0.44) KCNH2SLC2A1
SCHEMBL3375788 0.81 KCNH2 (0.44) KCNH2SLC2A1
SCHEMBL4792306 0.77 SLC2A1 (0.37) KCNH2SLC2A1
SCHEMBL3378451 0.74 KCNH2 (0.40) KCNH2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987040-B1 ETHANOL OR 1,2-ETHANEDIOL CYCLOHEXYL ANTIBIOTIC DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-11-10 EP claimed