SCHEMBL3376845

SCHEMBL3376845

CCOc1ccccc1C(=O)NC1CCCn2c1nc(-c1ccncc1)cc2=O

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 2/20 0.46
TSHR P16473 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HCRTR1 O43613 2/20 0.44
GSK3B P49841 2/20 0.44
USP2 O75604 2/20 0.44
KDM4D Q6B0I6 1/20 0.43
RXFP1 Q9HBX9 1/20 0.42
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.42
HTR7 P34969 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2064451 0.91 HCRTR2 (0.38) HCRTR2TSHRSMN1; SMN2HCRTR1GSK3B
SCHEMBL2065326 0.90 KMT2A (0.46) HCRTR2TSHRHCRTR1GSK3BKDM4D
SCHEMBL2064928 0.88 KDM5A (0.41) HCRTR2TSHRHCRTR1GSK3BKDM4D
SCHEMBL2065962 0.88 KMT2A (0.46) HCRTR2TSHRHCRTR1GSK3BKDM4D
SCHEMBL2064796 0.86 CGAS (0.39) GSK3BALDH1A1MEN1KMT2A
SCHEMBL2067036 0.86 CYP2C9 (0.40) HCRTR2HCRTR1GSK3B
SCHEMBL4383616 0.84 MEN1 (0.47) ALDH1A1MEN1KMT2A
SCHEMBL2066118 0.84 ALDH1A1 (0.43) HCRTR2HCRTR1GSK3BKDM4DALDH1A1
SCHEMBL2066786 0.83 GSK3B (0.47) HCRTR2HCRTR1GSK3BMEN1KMT2A
SCHEMBL4952879 0.82 MEN1 (0.47) ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957492-B1 SUBSTITUTED BICYCLIC PYRIMIDONE DERIVATIVES SANOFI AVENTIS (FR) 2010-11-10 EP claimed
EP-1957492-A2 SUBSTITUTED BICYCLIC PYRIMIDONE DERIVATIVES sanofi-aventis (FR) 2008-08-20 EP claimed
WO-2007057790-A2 SUBSTITUTED BICYCLIC PYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2007-05-24 WO claimed