SCHEMBL3378009

SCHEMBL3378009

O=C(N[C@H]1CCC[C@@](O)(C#Cc2cccc(Cl)c2)C1)Oc1ccoc1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 8/20 0.45
FAAH O00519 2/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 1/20 0.35
EPHX2 P34913 1/20 0.34
EPHX1 P07099 1/20 0.34
LHCGR P22888 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3374407 1.00 GRM5 (0.45) GRM5FAAHALDH1A1RAB9AEPHX2
SCHEMBL3841449 0.89 GRM5 (0.46) GRM5FAAHALDH1A1RAB9AEPHX2
SCHEMBL3841794 0.89 GRM5 (0.46) GRM5FAAHALDH1A1RAB9AEPHX2
SCHEMBL3374694 0.85 GRM5 (0.46) GRM5RAB9AEPHX2
SCHEMBL3374718 0.85 GRM5 (0.46) GRM5RAB9AEPHX2
SCHEMBL990758 0.84 GRM5 (0.45) GRM5RAB9A
SCHEMBL991434 0.84 GRM5 (0.45) GRM5RAB9A
SCHEMBL3374691 0.84 GRM5 (0.45) GRM5FAAHALDH1A1RAB9AEPHX2
SCHEMBL3374841 0.83 GRM5 (0.44) GRM5FAAHALDH1A1RAB9AEPHX2
SCHEMBL3374792 0.83 GRM5 (0.46) GRM5RAB9AEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877365-B1 ACETYLENE DERIVATIVES NOVARTIS AG (CH) 2010-11-10 EP claimed