SCHEMBL3378207

SCHEMBL3378207

COc1cc(F)c2nccc([C@@H](O)[C@H](O)[C@H]3CC[C@H](NC(=O)/C=C/c4cc(F)ccc4F)CC3)c2c1.COc1cc(F)c2nccc([C@@H](O)[C@H](O)[C@H]3CC[C@H](NC/C=C/c4cc(F)ccc4F)CC3)c2c1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 5/20 0.34
DRD2 P14416 3/20 0.34
DRD3 P35462 3/20 0.34
PTGS2 P35354 2/20 0.34
KCNH2 Q12809 2/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3377688 0.94 SLC2A1 (0.36) SLC2A1KCNH2
SCHEMBL3377820 0.94 SLC2A1 (0.36) SLC2A1KCNH2
SCHEMBL3377827 0.94 SLC2A1 (0.36) SLC2A1KCNH2
SCHEMBL3374581 0.94 PTGS2 (0.38) SLC2A1DRD2DRD3PTGS2KCNH2
SCHEMBL3376061 0.94 PTGS2 (0.38) SLC2A1DRD2DRD3PTGS2KCNH2
SCHEMBL3376066 0.94 PTGS2 (0.38) SLC2A1DRD2DRD3PTGS2KCNH2
SCHEMBL3376060 0.94 PTGS2 (0.38) SLC2A1DRD2DRD3PTGS2KCNH2
SCHEMBL3377824 0.94 SLC2A1 (0.36) SLC2A1KCNH2
SCHEMBL3378412 0.78 KCNH2 (0.51) SLC2A1KCNH2
SCHEMBL3378415 0.78 KCNH2 (0.51) SLC2A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987040-B1 ETHANOL OR 1,2-ETHANEDIOL CYCLOHEXYL ANTIBIOTIC DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-11-10 EP claimed