SCHEMBL3378372

SCHEMBL3378372

O=C(NC1CCCC1)Oc1cnc(Nc2ccc(Cl)cc2Cl)nc1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 9/20 0.53
RAB9A P51151 1/20 0.46
PTK2 Q05397 5/20 0.43
CYP3A4 P08684 4/20 0.43
CYP2C9 P11712 4/20 0.43
CYP1A2 P05177 4/20 0.43
LRRK2 Q5S007 3/20 0.43
CYP2C19 P33261 4/20 0.43
IGF1R P08069 1/20 0.41
CYP2D6 P10635 1/20 0.41
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3381212 0.98 CNR2 (0.53) CNR2RAB9APTK2CYP3A4CYP2C9
SCHEMBL3380132 0.91 CNR2 (0.53) CNR2PTK2CYP3A4CYP2C9CYP1A2
SCHEMBL3383470 0.86 CNR2 (0.64) CNR2CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL3381292 0.86 CNR2 (0.59) CNR2RAB9ACYP3A4CYP2C9CYP1A2
SCHEMBL3379863 0.85 CNR2 (0.63) CNR2CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL3382316 0.85 CNR2 (0.66) CNR2RAB9ACYP3A4CYP2C9CYP1A2
SCHEMBL3379589 0.84 CNR2 (0.52) CNR2PTK2CYP3A4CYP2C9CYP1A2
SCHEMBL3382862 0.84 CNR2 (0.59) CNR2PTK2CYP3A4CYP2C9CYP1A2
SCHEMBL3381376 0.84 CNR2 (0.66) CNR2CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL3380444 0.84 CNR2 (0.65) CNR2RAB9ACYP3A4CYP2C9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878725-B1 Pyrimidine derivatives and their use as CB2 modulators GLAXO GROUP LTD (GB) 2010-11-24 EP claimed