SCHEMBL33790

SCHEMBL33790

CC1(N)N=CN=C2N=CN=C21

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6897683 0.78
SCHEMBL8429764 0.77
SCHEMBL11346226 0.76
SCHEMBL3321079 0.75
SCHEMBL7118357 0.75
SCHEMBL157962 0.75
SCHEMBL17744967 0.75
SCHEMBL427042 0.71
SCHEMBL8885450 0.70
SCHEMBL9563447 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12104 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122071704-A SiRNA targeting bone morphogenetic protein 2, modified siRNA and application thereof 北京大学 2026-05-22 CN claimed
CN-122071703-A SiRNA targeting bone morphogenetic protein 4 gene, modified siRNA and application thereof 北京大学 2026-05-22 CN claimed
US-12630827-B2 Antisense oligonucleotides targeting SCN2A for the treatment of SCN1A encephalopathies ROGCON, INC. (US) 2026-05-19 US claimed
US-20260071273-A1 METHODS FOR NUCLEIC ACID SEQUENCING NANOHYB LLC (US) 2026-03-12 US claimed
EP-4705481-A2 CIRCULAR RNA COMPOSITIONS AND METHODS Orna Therapeutics, Inc. (US) 2026-03-11 EP claimed
EP-4677107-A1 METHOD FOR NATIVE STRAND SEQUENCING OF ENRICHED GENOMIC REGIONS Nanohyb, LLC (US) 2026-01-14 EP claimed
US-20250346624-A1 POLYNUCLEOTIDE AND PRODUCING METHOD THEREOF EISAI R&D MAN CO LTD (JP) 2025-11-13 US claimed
EP-4620970-A1 PORIN MONOMER, PORIN, MUTANT THEREOF, AND USE THEREOF BGI Shenzhen (CN) 2025-09-24 EP claimed
EP-4617375-A2 METHODS, COMPOSITIONS AND SYSTEMS FOR IMPROVING THE BINDING OF METHYLATED POLYNUCLEOTIDES Guardant Health, Inc. (US) 2025-09-17 EP claimed
EP-3821033-B1 USE OF DROPLET SINGLE CELL EPIGENOME PROFILING FOR PATIENT STRATIFICATION HIFIBIO SAS (FR) 2025-09-10 EP claimed
US-20020039741-A1 Antitumor agent DEAN NICHOLAS M (US) 2002-04-04 US claimed
EP-0957926-A4 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS FOR THE MODULATION OF THE EXPRESSION OF B7 PROTEIN ISIS PHARMACEUTICALS INC (US) 2002-01-23 EP claimed
US-6319906-B1 FOR THERAPY OF AUTOIMMUNE DISEASE, INFLAMMATORY DISEASE, FOR INHIBITING ALLOGRAFT REJECTION ISIS PHARMACEUTICALS 2001-11-20 US claimed
US-6312900-B1 FOR MODULATING METASTASIS OF MALIGNANT TUMORS VIA MODULATION OF ACTIVATING PROTEIN 1 ISIS PHARMACEUTICALS, INC. 2001-11-06 US claimed
JP-2000507833-A 2000-06-27 JP claimed
US-6077833-A FOR DIAGNOSIS, PREVENTION AND TREATMENT OF IMMUNE STATES AND DISORDERS AMENABLE TO TREATMENT THROUGH MODULATION OF T CELL ACTIVATION SUCH AS FOR PREVENTING ALLOGRAFT REJECTION ISIS PHARMACEUTICALS, INC. (US) 2000-06-20 US claimed
EP-0957926-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS FOR THE MODULATION OF THE EXPRESSION OF B7 PROTEIN ISIS PHARMACEUTICALS, INC. (US) 1999-11-24 EP claimed
US-5985558-A DNA SEQUENCE ISIS PHARMACEUTICALS INC. (US) 1999-11-16 US claimed
US-5837852-A PHOSPHORYLATED OLIGONUCLEOTIDE USE AS ANTIINFLUENZA AGENT, ENZYME INHIBITOR NOT DEPHOSPHORYLATED BY VIRAL POLYMERASE AND INHIBITORS OF INFLUENZA TRANSCRIPTION BRISTOL-MYERS SQUIBB COMPANY (US) 1998-11-17 US claimed
WO-1998029124-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS FOR THE MODULATION OF THE EXPRESSION OF B7 PROTEIN ISIS PHARMACEUTICALS, INC. (US) 1998-07-09 WO claimed