SCHEMBL3379141

SCHEMBL3379141

COc1cc2c(cc1NS(=O)(=O)O)CCC1C2CC[C@@]2(C)C1CC[C@@H]2OC

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 5/20 0.63
CA9 Q16790 5/20 0.63
STS P08842 8/20 0.59
CYP3A4 P08684 3/20 0.56
CYP1A2 P05177 2/20 0.56
HSD17B10 Q99714 2/20 0.56
CYP1A1 P04798 2/20 0.56
CYP1B1 Q16678 2/20 0.56
CYP19A1 P11511 2/20 0.56
TP53 P04637 2/20 0.56
MAPT P10636 2/20 0.56
TSHR P16473 1/20 0.56
NFKB1 P19838 1/20 0.56
CYP2C19 P33261 1/20 0.56
THPO P40225 1/20 0.56
MEN1 O00255 1/20 0.56
GMNN O75496 1/20 0.56
LMNA P02545 1/20 0.56
SHBG P04278 1/20 0.56
GAA P10253 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3379139 1.00 CA2 (0.63) CA2CA9STSCYP3A4CYP1A2
SCHEMBL3381694 0.90 STS (0.58) CA2CA9STSCYP3A4TP53
SCHEMBL3381697 0.90 STS (0.58) CA2CA9STSCYP3A4TP53
SCHEMBL5265236 0.90 STS (0.70) CA2CA9STSCYP3A4CYP1A2
SCHEMBL6639220 0.90 STS (0.70) CA2CA9STSCYP3A4CYP1A2
SCHEMBL3378635 0.90 CA2 (0.58) CA2CA9STSCYP3A4CYP1A2
SCHEMBL3378639 0.90 CA2 (0.58) CA2CA9STSCYP3A4CYP1A2
SCHEMBL5265240 0.90 STS (0.70) CA2CA9STSCYP3A4CYP1A2
SCHEMBL5265994 0.90 STS (0.70) CA2CA9STSCYP3A4CYP1A2
SCHEMBL5265990 0.90 STS (0.70) CA2CA9STSCYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599493-B1 2-SUBSTITUTED ESTRA-1,3,5(10)-TRIENE-3-YL SULFAMATE WITH AN ANTI-TUMOUR ACTION STERIX LTD (GB) 2010-11-24 EP claimed