SCHEMBL3379218

SCHEMBL3379218

O=C(Nc1ccccc1)Oc1cccc2c1Oc1ccccc1C2=C1CC2CCC(C1)N2

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
HSP90AA1 P07900 1/20 0.36
LMNA P02545 1/20 0.34
MC4R P32245 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3382988 0.86 HTR1A (0.41) ALDH1A1KDM4ELMNABCHE
SCHEMBL3381652 0.85 CHRNA7 (0.33)
SCHEMBL3382426 0.83 CHRNA7 (0.32)
SCHEMBL3382541 0.83 CREBBP (0.42) ALDH1A1KDM4EKMT2ALMNA
SCHEMBL3384341 0.78 CHRNA7 (0.36) ALDH1A1KMT2AHSP90AA1LMNA
SCHEMBL3384638 0.77 KDM4E (0.32) GAAALDH1A1KDM4EKMT2A
SCHEMBL3383083 0.75 SETD7 (0.35)
SCHEMBL3384775 0.74 BRD4 (0.37) GAA
Trifluoroacetic Acid SCHEMBL3382424 0.73 KDM1A (0.36)
SCHEMBL4669628 0.73 SETD7 (0.46) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896467-B1 TRICYCLIC OPIOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2010-12-01 EP claimed