SCHEMBL3379226

SCHEMBL3379226

N#Cc1cccc(Nc2ncc(OC(=O)NCC3CCCCC3)c(C(F)(F)F)n2)c1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 14/20 0.57
CYP2C19 P33261 5/20 0.57
CYP3A4 P08684 4/20 0.57
CYP2C9 P11712 4/20 0.57
CYP1A2 P05177 4/20 0.55
CYP2D6 P10635 3/20 0.53
MAOB P27338 1/20 0.44
GRM5 P41594 1/20 0.44
TSHR P16473 1/20 0.43
SYK P43405 2/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3382370 0.99 CNR2 (0.56) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3382339 0.92 CNR2 (0.58) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3381193 0.90 CNR2 (0.50) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3382877 0.89 CNR2 (0.51) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3380608 0.88 CNR2 (0.60) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3383239 0.87 CNR2 (0.74) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3380187 0.87 CNR2 (0.59) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3382577 0.87 CNR2 (0.59) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3380875 0.87 CNR2 (0.57) CNR2CYP2C19CYP3A4CYP2C9CYP1A2
SCHEMBL3381115 0.86 CNR2 (0.59) CNR2CYP2C19CYP3A4CYP2C9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878725-B1 Pyrimidine derivatives and their use as CB2 modulators GLAXO GROUP LTD (GB) 2010-11-24 EP claimed