SCHEMBL3379565

SCHEMBL3379565

O=C(O)C[C@H]1CCCc2c1cnn2-c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.58
TMEM97 Q5BJF2 1/20 0.58
DHODH Q02127 6/20 0.49
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
USP30 Q70CQ3 1/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3378446 1.00 SIGMAR1 (0.58) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL955851 1.00 SIGMAR1 (0.58) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL8443811 0.87 TMEM97 (0.53) SIGMAR1TMEM97DHODHKMT2A
SCHEMBL959673 0.86 TMEM97 (0.55) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL8443685 0.85 TMEM97 (0.52) SIGMAR1TMEM97DHODH
SCHEMBL9276021 0.85 TMEM97 (0.52) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL9282253 0.85 TMEM97 (0.52) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL9282677 0.85 TMEM97 (0.52) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL958122 0.85 TMEM97 (0.52) SIGMAR1TMEM97DHODH
SCHEMBL956196 0.84 SIGMAR1 (0.67) SIGMAR1TMEM97DHODHKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010066829-A1 PROCESS FOR OBTAINING ENANTIOMERICALLY ENRICHED PYRAZOLE DERIVATIVES LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2010-06-17 WO disclosed
WO-2010066829-A1 PROCESS FOR OBTAINING ENANTIOMERICALLY ENRICHED PYRAZOLE DERIVATIVES LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2010-06-17 WO disclosed
EP-2196458-A1 Process for obtaining enantiomerically enriched pyrazole derivatives Laboratorios Del. Dr. Esteve, S.A. (ES) 2010-06-16 EP disclosed
EP-2196458-A1 Process for obtaining enantiomerically enriched pyrazole derivatives Laboratorios Del. Dr. Esteve, S.A. (ES) 2010-06-16 EP disclosed