SCHEMBL3382008

SCHEMBL3382008

O=C(O)N1Cc2cc(Cl)ccc2-n2c(nnc2[C@H]2CC[C@H](Oc3ccc4ccccc4c3)CC2)C1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 18/20 0.55
KCNH2 Q12809 9/20 0.55
AVPR2 P30518 8/20 0.55
OXTR P30559 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15233987 0.92 AVPR1A (0.59) AVPR1AKCNH2AVPR2OXTR
SCHEMBL15234146 0.92 AVPR1A (0.59) AVPR1AKCNH2AVPR2OXTR
SCHEMBL15234203 0.91 AVPR1A (0.56) AVPR1AKCNH2AVPR2OXTR
SCHEMBL3330454 0.89 AVPR1A (0.56) AVPR1AKCNH2AVPR2OXTR
SCHEMBL15234220 0.88 OXTR (0.58) AVPR1AKCNH2AVPR2OXTR
SCHEMBL15234244 0.87 AVPR1A (0.55) AVPR1AKCNH2AVPR2OXTR
SCHEMBL15234246 0.87 AVPR1A (0.55) AVPR1AKCNH2AVPR2OXTR
SCHEMBL3379061 0.87 AVPR1A (0.55) AVPR1AKCNH2AVPR2OXTR
SCHEMBL3327242 0.87 AVPR1A (0.64) AVPR1AKCNH2AVPR2OXTR
SCHEMBL15234093 0.86 AVPR1A (0.51) AVPR1AKCNH2AVPR2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010060836-A1 ARYLCYCLOHEXYLETHERS OF DIHYDROTETRAAZABENZOAZULENES FOR USE AS VASOPRESSIN VIA RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-06-03 WO claimed