SCHEMBL3383547

SCHEMBL3383547

CC(C)(C)c1cc(NC(=O)Cc2ccc(-c3cnc4cc(-c5ccnc(F)c5)ccn34)cc2)no1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RET P07949 12/20 0.56
NTRK1 P04629 3/20 0.48
CSF1R P07333 1/20 0.47
KDR P35968 1/20 0.47
KCNH2 Q12809 1/20 0.47
CCDC6 Q16204 1/20 0.47
WNT3A P56704 4/20 0.46
ROCK1 Q13464 1/20 0.46
FLT3 P36888 1/20 0.42
KIT P10721 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3385345 0.91 RET (0.60) RETNTRK1CSF1RKDRKCNH2
SCHEMBL3386505 0.85 RET (0.65) RETNTRK1CSF1RKDRKCNH2
SCHEMBL3176763 0.85 RET (0.53) RETNTRK1CSF1RKDRKCNH2
SCHEMBL3188885 0.85 RET (0.58) RETNTRK1CSF1RKDRKCNH2
SCHEMBL3383110 0.82 RET (0.48) RETNTRK1CSF1RKDRKCNH2
SCHEMBL3186841 0.82 RET (0.53) RETNTRK1CSF1RKDRKCNH2
SCHEMBL3185001 0.81 RET (0.52) RETNTRK1CSF1RKDRKCNH2
SCHEMBL3178793 0.80 RET (0.51) RETNTRK1CSF1RKDRKCNH2
SCHEMBL3385534 0.79 KDR (0.50) RETKDRFLT3
SCHEMBL3383013 0.79 RET (0.48) RETNTRK1CSF1RKDRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed