SCHEMBL3384064

SCHEMBL3384064

O=C(NCc1ccc(-c2cnc3cc(-c4ccsc4)ccn23)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
FGFR3 P22607 17/20 0.48
KDR P35968 17/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3384511 0.86 KDR (0.55) FGFR3KDR
SCHEMBL3384065 0.79 KDR (0.52) FGFR3KDR
SCHEMBL3381138 0.77 KDR (0.42) FGFR3KDR
SCHEMBL11929274 0.76 FGFR3 (0.79) FGFR3KDR
SCHEMBL3383984 0.75 KDR (0.68) FGFR3KDR
SCHEMBL3380720 0.75 KDR (0.58) FGFR3KDR
SCHEMBL3385738 0.74 FLT3 (0.49) FGFR3KDR
SCHEMBL27705887 0.74 FGFR3 (0.54) FGFR3KDR
SCHEMBL1790420 0.74 CA1 (0.67) CA1CA2CA7CA9KDR
SCHEMBL3177632 0.74 FGFR3 (0.56) FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128461-B Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI 2010-12-22 CN disclosed
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed