SCHEMBL3384065

SCHEMBL3384065

O=C(Cc1ccc(-c2cnc3cc(-c4ccncc4)ccn23)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 0.52
FGFR3 P22607 7/20 0.52
BLM P54132 1/20 0.45
BRAF P15056 1/20 0.45
PLA2G7 Q13093 1/20 0.45
FLT1 P17948 3/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
KCNJ5 P48544 1/20 0.44
KCNJ3 P48549 1/20 0.44
GRM4 Q14833 1/20 0.43
CSF1R P07333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3385738 0.89 FLT3 (0.49) KDRFGFR3MEN1KMT2AMAPT
SCHEMBL13483163 0.88 FGFR3 (0.50) KDRFGFR3BLM
SCHEMBL3195980 0.85 RET (0.60) KDRFGFR3MEN1KMT2AMAPT
SCHEMBL3385496 0.80 KDR (0.50) KDRFGFR3MEN1KMT2A
SCHEMBL3385476 0.79 KDR (0.49) KDRFGFR3FLT1CSF1R
SCHEMBL3384064 0.79 CA1 (0.49) KDRFGFR3
SCHEMBL3382028 0.78 KDR (0.58) KDRFGFR3
SCHEMBL3417117 0.78 WNT3A (0.49) KDRFGFR3
SCHEMBL3381109 0.77 RET (0.56) KDRFGFR3
SCHEMBL3384190 0.76 KDR (0.62) KDRFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128461-B Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI 2010-12-22 CN disclosed
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed
CN-101128461-A Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI (US) 2008-02-20 CN disclosed