SCHEMBL3384506

SCHEMBL3384506

O=C(Cc1ccc(-c2cnc3cc(-c4ccncc4)ccn23)cc1F)Nc1cccc(C(F)(F)F)c1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.59
FGFR3 P22607 12/20 0.59
DDR1 Q08345 4/20 0.51
DDR2 Q16832 4/20 0.51
ABL1 P00519 3/20 0.51
BCR P11274 3/20 0.51
KIT P10721 2/20 0.51
RET P07949 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3184828 0.93 KDR (0.55) KDRFGFR3DDR1DDR2ABL1
SCHEMBL3381852 0.93 KDR (0.56) KDRFGFR3DDR1
SCHEMBL3188712 0.91 DDR1 (0.52) KDRFGFR3DDR1DDR2ABL1
SCHEMBL3382028 0.91 KDR (0.58) KDRFGFR3DDR1DDR2ABL1
SCHEMBL3183878 0.91 KDR (0.54) KDRFGFR3
SCHEMBL3383795 0.89 KDR (0.60) KDRFGFR3DDR1DDR2ABL1
SCHEMBL3195980 0.88 RET (0.60) KDRFGFR3DDR1DDR2ABL1
SCHEMBL3385818 0.88 KDR (0.49) KDRFGFR3DDR1DDR2ABL1
SCHEMBL3383730 0.88 FGFR3 (0.55) KDRFGFR3
SCHEMBL3385328 0.87 FGFR3 (0.55) KDRFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128461-B Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI 2010-12-22 CN disclosed
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed
CN-101128461-A Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI (US) 2008-02-20 CN disclosed