SCHEMBL3385328

SCHEMBL3385328

CC(C)(C)C(=O)c1cccc(NC(=O)Cc2ccc(-c3cnc4cc(-c5ccncc5)ccn34)cc2F)c1

nearest known ligand 0.55

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 19/20 0.55
KDR P35968 19/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3383730 0.93 FGFR3 (0.55) FGFR3KDR
SCHEMBL3381852 0.90 KDR (0.56) FGFR3KDR
SCHEMBL3184828 0.88 KDR (0.55) FGFR3KDR
SCHEMBL3183878 0.88 KDR (0.54) FGFR3KDR
SCHEMBL3384506 0.87 KDR (0.59) FGFR3KDR
SCHEMBL3187558 0.84 FGFR3 (0.50) FGFR3KDR
SCHEMBL3382504 0.81 KDR (0.47) FGFR3KDR
SCHEMBL3188712 0.81 DDR1 (0.52) FGFR3KDR
SCHEMBL3380938 0.80 KDR (0.46) FGFR3KDR
SCHEMBL3383110 0.80 RET (0.48) FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128461-B Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI 2010-12-22 CN disclosed
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed
CN-101128461-A Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI (US) 2008-02-20 CN disclosed