SCHEMBL3386535

SCHEMBL3386535

CC(C)(C)[Si](C)(C)O[C@@H](CN)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.41
HTR2A P28223 1/20 0.41
CHRNB2 P17787 3/20 0.41
CHRNA4 P43681 3/20 0.41
SLC6A2 P23975 3/20 0.40
SLC6A4 P31645 3/20 0.40
SLC6A3 Q01959 3/20 0.40
NOS2 P35228 1/20 0.39
CA2 P00918 1/20 0.36
AOC3 Q16853 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386613 1.00 TAAR1 (0.41) TAAR1HTR2ACHRNB2CHRNA4SLC6A2
SCHEMBL3386536 1.00 TAAR1 (0.41) TAAR1HTR2ACHRNB2CHRNA4SLC6A2
SCHEMBL23354701 0.85 CA2 (0.35) CA2
SCHEMBL23354817 0.83 CFTR (0.38) SLC6A2SLC6A4SLC6A3CA2
SCHEMBL8405099 0.83 GSR (0.44) SLC6A2SLC6A4SLC6A3CA2AOC3
SCHEMBL14984000 0.83 GSR (0.44) SLC6A2SLC6A4SLC6A3CA2AOC3
SCHEMBL1739510 0.83 GSR (0.44) SLC6A2SLC6A4SLC6A3CA2AOC3
SCHEMBL7151617 0.82 TAAR1 (0.47) TAAR1HTR2ACHRNB2CHRNA4SLC6A2
SCHEMBL9626551 0.82 TAAR1 (0.47) TAAR1HTR2ACHRNB2CHRNA4SLC6A2
SCHEMBL7392343 0.82 AOC3 (0.46) CHRNB2CHRNA4SLC6A4NOS2CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3548465-A1 THIONYL TETRAFLUORIDE MODIFIED COMPOUNDS AND USES The Scripps Research Institute (US) 2019-10-09 EP disclosed
WO-2018102433-A1 THIONYL TETRAFLUORIDE MODIFIED COMPOUNDS AND USES THE SCRIPPS RESEARCH INSTITUTE (US) 2018-06-07 WO disclosed
EP-1864995-B1 BETA-LACTAMIC RGD CYCLOPEPTIDES CONTAINING GAMMA TURNS UNIV PAIS VASCO (ES) 2010-12-08 EP disclosed
EP-1864995-A1 BETA-LACTAMIC RGD CYCLOPEPTIDES CONTAINING GAMMA TURNS UNIVERSIDAD DEL PAIS VASCO-EUSKAL HERRIKO UNIBERSITATEA (ES) 2007-12-12 EP disclosed
US-20030143701-A1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEMICAL INDUSTRIES, LTD. 2003-07-31 US disclosed
EP-0924194-B1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEM (JP) 2003-05-14 EP disclosed
US-6528686-B1 Reacting primary amine and ketone functionalized derivatives; catalytically reducing DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2003-03-04 US disclosed
EP-0924193-B1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEM (JP) 2003-02-19 EP disclosed
EP-0939134-B1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEM (JP) 2002-09-11 EP disclosed
US-6114582-A DECYCLIZATION TO FORM A CHEMICAL INTERMEDIATE FOR PRODUCING AN ANTI-OBESITY AGENT AND ANTIDIABETIC AGENT DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-05 US disclosed
EP-0654534-B1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEM (JP) 2000-03-01 EP disclosed
EP-0939134-A1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-09-01 EP disclosed
EP-0924194-A2 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-06-23 EP disclosed
EP-0924193-A1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-06-23 EP disclosed
US-5811293-A CULTURE PRODUCT AS CHEMICAL INTERMEDIATE FOR ANTI-OBESITY AGENT DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-22 US disclosed
US-5629200-A MICROORGANISM DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-13 US disclosed
EP-0654534-A2 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1995-05-24 EP disclosed