SCHEMBL3386793

SCHEMBL3386793

NC(Cc1cccc(C(F)(F)F)c1)c1nc(O)c2cc(-c3cn[nH]c3)ccc2n1

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 17/20 0.68
ROCK1 Q13464 3/20 0.46
AKT1 P31749 2/20 0.43
PRKACA P17612 1/20 0.43
PRKACG P22612 1/20 0.43
PRKACB P22694 1/20 0.43
NPBWR1 P48145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386790 1.00 ROCK2 (0.68) ROCK2ROCK1AKT1PRKACAPRKACG
SCHEMBL3389658 0.88 ROCK2 (0.75) ROCK2ROCK1
SCHEMBL3386619 0.88 ROCK2 (0.75) ROCK2ROCK1
SCHEMBL3386625 0.88 ROCK2 (0.75) ROCK2ROCK1
SCHEMBL3383157 0.88 ROCK2 (0.63) ROCK2ROCK1
SCHEMBL3383164 0.88 ROCK2 (0.63) ROCK2ROCK1
SCHEMBL3387757 0.86 ROCK2 (0.67) ROCK2ROCK1
SCHEMBL3387761 0.86 ROCK2 (0.67) ROCK2ROCK1
SCHEMBL3387576 0.83 ROCK2 (0.66) ROCK2ROCK1
SCHEMBL3387565 0.83 ROCK2 (0.66) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010056758-A1 QUINAZOLINE DERIVATIVES AS KINASE INHIBITORS FENG YANGBO (US) 2010-05-20 WO disclosed