SCHEMBL3387133

SCHEMBL3387133

CC(O)Nc1nc(NCc2ccccn2)c2c(-c3ccc(F)cc3)csc2n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 5/20 0.52
TNF P01375 2/20 0.52
NOD1 Q9Y239 2/20 0.52
KCNA5 P22460 5/20 0.47
PIP4K2C Q8TBX8 1/20 0.44
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
PKM P14618 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NPR1 P16066 1/20 0.42
KCNH2 Q12809 5/20 0.41
CCNE1 P24864 8/20 0.40
CDK2 P24941 8/20 0.40
CDK4 P11802 7/20 0.40
CCND1 P24385 7/20 0.40
CDK7 P50613 7/20 0.40
CCNH P51946 7/20 0.40
CDK1 P06493 6/20 0.40
CCNB1 P14635 6/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2368786 0.88 TNF (0.57) MAPK1TNFNOD1KCNA5PIP4K2C
SCHEMBL2368804 0.86 TNF (0.55) MAPK1TNFNOD1KCNA5PIP4K2C
SCHEMBL27660750 0.85 TNF (0.64) MAPK1TNFNOD1KCNA5PIP4K2C
SCHEMBL3386735 0.84 TNF (0.59) MAPK1TNFNOD1KCNA5PIP4K2C
SCHEMBL2369487 0.83 TNF (0.52) MAPK1TNFNOD1KCNA5PIP4K2C
SCHEMBL2368704 0.83 MAPK1 (0.64) MAPK1TNFNOD1KCNA5PIP4K2C
SCHEMBL2369260 0.82 TNF (0.55) MAPK1TNFNOD1KCNA5PIP4K2C
SCHEMBL2368795 0.82 TNF (0.59) MAPK1TNFNOD1KCNA5PIP4K2C
SCHEMBL3385334 0.82 ESR1 (0.61) MAPK1TNFNOD1KCNA5PIP4K2C
SCHEMBL3384953 0.81 KCNH2 (0.57) MAPK1TNFNOD1KCNA5PIP4K2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641803-B3 THIENOPYRIMIDINE DERIVATIVES AS POTASSIUM CHANNEL INHIBITORS XENTION LTD (GB) 2010-12-08 EP disclosed