SCHEMBL3387481

SCHEMBL3387481

CC(C)(C)OC(=O)ON1CCC(Nc2nc(N)c(C(=O)c3cccc(F)c3)s2)CC1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 10/20 0.65
CDK5R1 Q15078 10/20 0.65
CCNA2 P20248 8/20 0.59
CDK2 P24941 8/20 0.59
KDM4E B2RXH2 1/20 0.42
TP53 P04637 1/20 0.42
HTT P42858 1/20 0.42
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HIF1A Q16665 1/20 0.42
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27686737 0.92 CDK5 (0.68) CDK5CDK5R1CCNA2CDK2KDM4E
SCHEMBL3384712 0.89 CCNA2 (0.74) CDK5CDK5R1CCNA2CDK2
SCHEMBL3389650 0.86 CCNA2 (0.53) CDK5CDK5R1CCNA2CDK2KDM4E
SCHEMBL3386774 0.83 CDK5 (0.72) CDK5CDK5R1CCNA2CDK2KDM4E
SCHEMBL3386683 0.82 CDK5 (0.74) CDK5CDK5R1CCNA2CDK2
SCHEMBL3384847 0.81 CDK5 (0.70) CDK5CDK5R1CCNA2CDK2
SCHEMBL28765719 0.81 CDK5 (0.67) CDK5CDK5R1CCNA2CDK2KDM4E
SCHEMBL28765718 0.81 CDK5 (0.69) CDK5CDK5R1CCNA2CDK2KDM4E
SCHEMBL3389148 0.79 CDK2 (0.49) CDK5CDK5R1CCNA2CDK2GSK3A
SCHEMBL14073849 0.79 CDK5 (0.67) CDK5CDK5R1CCNA2CDK2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771424-B1 NOVEL 2,4-DIAMINOTHIAZOL-5-ONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-12-15 EP claimed