SCHEMBL3387770

SCHEMBL3387770

Cc1cnc2cc(-c3cccc(CN4CCCCC4)c3)ccc2n1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.51
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48
CNR2 P34972 3/20 0.47
CNR1 P21554 2/20 0.47
HDAC6 Q9UBN7 1/20 0.46
KDM5B Q9UGL1 1/20 0.45
S1PR1 P21453 1/20 0.45
AVPR1B P47901 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
TDP1 Q9NUW8 1/20 0.45
ALDH1A1 P00352 1/20 0.45
PDE2A O00408 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44
BACE1 P56817 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24495604 0.76 CYP2D6 (0.62) HRH3CYP2D6CYP2C19SMN1; SMN2TDP1
SCHEMBL3432734 0.75 HRH3 (0.47) HRH3CYP2D6CYP2C19CNR2CNR1
SCHEMBL24495602 0.74 HRH3 (0.57) HRH3CYP2D6CYP2C19SMN1; SMN2TDP1
SCHEMBL3435319 0.74 HRH3 (0.46) HRH3CYP2D6CYP2C19CNR2CNR1
SCHEMBL22310287 0.74 S1PR1 (0.50) HRH3CYP2D6CYP2C19CNR2CNR1
SCHEMBL23440312 0.74 CYP2D6 (0.68) HRH3CYP2D6CYP2C19SMN1; SMN2TDP1
SCHEMBL12597039 0.74 CCNB2 (0.51) SMN1; SMN2ALDH1A1
SCHEMBL11992422 0.73 PRMT6 (0.48) HRH3CYP2D6CYP2C19CNR2CNR1
SCHEMBL3425973 0.72 CYP2D6 (0.65) HRH3CYP2D6CYP2C19SMN1; SMN2TDP1
SCHEMBL30572548 0.72 DHODH (0.68) CNR2CNR1HDAC6SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010052448-A2 FUSED PYRAZINE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2010-05-14 WO disclosed