SCHEMBL3388657

SCHEMBL3388657

O=C(c1ccc2[nH]ccc2c1)N1CCN(C2CCC2)CC1.O=C(c1ccc2c(ccn2C2CCN(Cc3ccccc3)C2)c1)N1CCN(C2CCC2)CC1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.60
CCR3 P51677 2/20 0.49
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 3/20 0.49
ACHE P22303 1/20 0.49
HTR4 Q13639 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
CHRM2 P08172 1/20 0.46
HRH3 Q9Y5N1 2/20 0.46
KMT2A Q03164 1/20 0.46
ACACB O00763 1/20 0.43
ACACA Q13085 1/20 0.43
NPC1 O15118 1/20 0.42
MBTD1 Q05BQ5 1/20 0.42
L3MBTL3 Q96JM7 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
OXTR P30559 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3390277 0.98 MAPK14 (0.60) MAPK14CCR3KDM4EALDH1A1ACHE
SCHEMBL3383892 0.94 MAPK14 (0.64) MAPK14CCR3KDM4EALDH1A1ACHE
SCHEMBL3387943 0.92 KDM4E (0.56) KDM4EALDH1A1ACHEHRH3KMT2A
SCHEMBL3388648 0.90 KDM4E (0.56) KDM4EALDH1A1ACHEHRH3KMT2A
SCHEMBL3391056 0.89 MAPK14 (0.59) MAPK14CCR3KDM4EALDH1A1ACHE
SCHEMBL3390881 0.89 MAPK14 (0.59) MAPK14CCR3KDM4EALDH1A1ACHE
SCHEMBL3390449 0.87 MAPK14 (0.57) MAPK14CCR3KDM4EACHEHTR4
SCHEMBL3387912 0.85 KDM4E (0.60) MAPK14KDM4EALDH1A1ACHEHRH3
SCHEMBL3388485 0.85 MAPK14 (0.56) MAPK14CCR3KDM4EALDH1A1ACHE
SCHEMBL3387677 0.84 MAPK14 (0.56) MAPK14CCR3KDM4EALDH1A1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029534-B1 1H-INDOL-5-YL-PIPERAZIN-1-YL-METHANONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-12-22 EP disclosed