Norketamine

Norketamine

SCHEMBL3390132

NC1(c2ccccc2Cl)CCCCC1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 3/20 0.59
GRIN2A Q12879 3/20 0.59
SLC6A4 P31645 2/20 0.59
GRIN2D O15399 2/20 0.59
GRIN3B O60391 2/20 0.59
GRIN2B Q13224 2/20 0.59
GRIN2C Q14957 2/20 0.59
GRIN3A Q8TCU5 2/20 0.59
OPRK1 P41145 1/20 0.59
LMNA P02545 1/20 0.59
OPRM1 P35372 1/20 0.59
CACNA1C Q13936 1/20 0.59
HDAC4 P56524 1/20 0.47
TSHR P16473 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Norketamine SCHEMBL30089863 1.00 GRIN1 (0.59) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
Norketamine SCHEMBL12601750 1.00 GRIN1 (0.59) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
Norketamine SCHEMBL30089862 1.00 GRIN1 (0.59) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
Norketamine SCHEMBL12601748 1.00 GRIN1 (0.59) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
Norketamine SCHEMBL30714777 1.00 GRIN1 (0.59) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
Norketamine SCHEMBL30546347 0.98 GRIN1 (0.57) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
Norketamine SCHEMBL29626880 0.98 GRIN1 (0.57) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
Norketamine SCHEMBL29626917 0.98 GRIN1 (0.57) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
SCHEMBL21452531 0.98 GRIN1 (0.57) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
Norketamine SCHEMBL1997948 0.98 GRIN1 (0.57) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 371 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3946296-B9 EXTENDED RELEASE PHARMACEUTICAL FORMULATION DOUGLAS PHARMACEUTICALS LTD (NZ) 2024-12-25 EP claimed
EP-3946296-B1 EXTENDED RELEASE PHARMACEUTICAL FORMULATION DOUGLAS PHARMACEUTICALS LTD (NZ) 2024-05-01 EP claimed
CN-114716332-B Preparation method of ketamine 宜昌人福药业有限责任公司 2023-06-02 CN claimed
US-20230000797-A1 COMPOSITIONS AND METHODS FOR TREATING MOTOR DISORDERS ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA 2023-01-05 US claimed
US-20220401366-A1 LONG ACTING NMDA ANTAGONISTS CONSEGNA PHARMA INC (US) 2022-12-22 US claimed
US-20220378777-A1 COMPOSITIONS AND METHODS FOR TREATING ALCOHOL USE DISORDER OR A RELATED CONDITION THEREOF THE TRUSTEES OF INDIANA UNIVERSITY 2022-12-01 US claimed
EP-3891505-B1 A METHOD FOR MEASURING A CONCENTRATION OF A BIOMARKER/ANALYTE IN BLOOD FROM MAMMALS REDHOTDIAGNOSTICS AB (SE) 2022-11-30 EP claimed
US-11426366-B2 Compositions and methods for treating motor disorders ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSSITY OF ARIZONA (US) 2022-08-30 US claimed
CN-114716332-A Preparation method of ketamine 宜昌人福药业有限责任公司 2022-07-08 CN claimed
WO-2021108801-A2 LONG ACTING NMDA ANTAGONISTS CONSEGNA PHARMA, INC. (US) 2021-06-03 WO claimed
WO-2021087258-A1 COMPOSITIONS AND METHODS FOR TREATING ALCOHOL USE DISORDER OR A RELATED CONDITION THEREOF THE TRUSTEES OF INDIANA UNIVERSITY (US) 2021-05-06 WO claimed
CN-110818587-A Preparation method of ketamine and synthesis method of intermediate compound 宜昌人福药业有限责任公司 2020-02-21 CN claimed
CN-122070289-A Hydroxynorketamine analogues and uses thereof 灵飞制药公司 2026-05-19 CN disclosed
US-20260130869-A1 ORAL DOSAGE FORM OF KETAMINE KETABON GMBH (DE) 2026-05-14 US disclosed
US-12611386-B2 Extended release pharmaceutical formulation DOUGLAS PHARMACEUTICALS LTD. (NZ) 2026-04-28 US disclosed
US-20260109663-A1 NEURO-ATTENUATING KETAMINE AND NORKETAMINE COMPOUNDS, DERIVATIVES THEREOF, AND METHODS ACADIA PHARM INC (US) 2026-04-23 US disclosed
EP-1333023-A1 Haptens, immunogens, antibodies and conjugates to ketamine and its metabolites Randox Laboratories Ltd. (GB) 2003-08-06 EP disclosed
US-5384331-A Ketamine analogues for treatment of thrombocytopenia GENENTECH, INC. (US) 1995-01-24 US disclosed
EP-0623343-A1 Ketamine analogues for the treatment of thrombocytopenia GENENTECH, INC. (US) 1994-11-09 EP disclosed
US-5250732-A Influence replication, differentiation or maturation of platelet progenitor cells GENENTECH, INC. (US) 1993-10-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230000797-A1 COMPOSITIONS AND METHODS FOR TREATING MOTOR DISORDERS SNCA, PARK7, COMT GRIN1 77/4885GRIN2A 38/4885SLC6A4 138/4885
US-20260109663-A1 NEURO-ATTENUATING KETAMINE AND NORKETAMINE COMPOUNDS, DERIVATIVES THEREOF, AND METHODS SLC6A4, KCNK4, KCNJ11 GRIN1 82/4885GRIN2A 116/4885SLC6A4 1/4885
US-20260130869-A1 ORAL DOSAGE FORM OF KETAMINE KCNQ2, KCNQ1, KCNQ3 GRIN1 122/4885GRIN2A 125/4885SLC6A4 315/4885
US-12611386-B2 Extended release pharmaceutical formulation HTR1D, GRIN1, GRIN2D GRIN1 2/4885GRIN2A 7/4885SLC6A4 16/4885
US-11426366-B2 Compositions and methods for treating motor disorders COMT, SNCA, PARK7 GRIN1 86/4885GRIN2A 40/4885SLC6A4 144/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.