Bicarbonate

Bicarbonate

SCHEMBL3391320

COc1cc(-c2ccc(Nc3nc4ccc(F)cc4s3)c(F)c2)ccc1C(=O)NC1CC1.O=C(O)O

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 2/20 0.56
HCRTR1 O43613 13/20 0.54
HCRTR2 O43614 8/20 0.54
MAPT P10636 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
SMYD3 Q9H7B4 1/20 0.46
GAK O14976 1/20 0.45
KMT2A Q03164 2/20 0.45
CLK1 P49759 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
TNF P01375 1/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
NR2F2 P24468 1/20 0.45
HTT P42858 1/20 0.45
MCL1 Q07820 1/20 0.45
KLF5 Q13887 1/20 0.45
NOD1 Q9Y239 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1761376 0.87 DGAT1 (0.56) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2
Bicarbonate SCHEMBL3386226 0.85 DGAT1 (0.69) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2
SCHEMBL1761337 0.85 MAPT (0.57) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2
SCHEMBL1761447 0.85 DGAT1 (0.51) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2
SCHEMBL1761521 0.83 DGAT1 (0.61) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2
SCHEMBL1761573 0.82 DGAT1 (0.49) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2
SCHEMBL1761387 0.82 DGAT1 (0.49) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2
Bicarbonate SCHEMBL3391760 0.82 DGAT1 (0.70) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2
SCHEMBL12593973 0.81 DGAT1 (0.52) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2
SCHEMBL1761410 0.81 DGAT1 (0.48) DGAT1HCRTR1HCRTR2MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805156-B1 PREPARATION AND USE OF BIPHENYL-4-YL-CARBONYLAMINO ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2010-12-22 EP claimed