SCHEMBL3393337

SCHEMBL3393337

N#Cc1ccc(-c2ccnc(NCc3cc(-c4ccccn4)[nH]n3)c2)c(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.58
TGFBR1 P36897 1/20 0.42
GRM5 P41594 3/20 0.39
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
CHEK1 O14757 1/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
CLK4 Q9HAZ1 2/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PDE5A O76074 2/20 0.37
LMNA P02545 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
MET P08581 1/20 0.36
IDH1 O75874 1/20 0.36
CRHR1 P34998 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13426080 0.89 KCNH2 (0.58) KCNH2ABCB1ABCG2CHEK1CYP1A2
SCHEMBL3392059 0.89 KCNH2 (0.74) KCNH2TGFBR1GRM5ABCB1ABCG2
SCHEMBL13426073 0.87 KCNH2 (0.46) KCNH2TGFBR1GRM5CYP1A2CYP2C19
SCHEMBL13426140 0.86 KCNH2 (0.49) KCNH2CYP1A2CYP2C19CLK4ALDH1A1
SCHEMBL13426213 0.86 KCNH2 (0.56) KCNH2TGFBR1ABCB1ABCG2CHEK1
SCHEMBL3393138 0.84 KCNH2 (0.50) KCNH2ABCB1ABCG2CYP1A2CYP2C19
SCHEMBL13426284 0.84 KCNH2 (0.59) KCNH2TGFBR1GRM5ABCB1ABCG2
SCHEMBL3395596 0.81 KCNH2 (0.40) KCNH2TGFBR1GRM5ABCB1ABCG2
SCHEMBL13425745 0.80 KCNH2 (0.60) KCNH2CYP1A2CYP2C19CLK4USP2
SCHEMBL13425826 0.80 KCNH2 (0.64) KCNH2CHEK1CYP1A2CYP2C19CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed