SCHEMBL3394056

SCHEMBL3394056

COc1ccc(C=Cc2cccc(O)c2)cc1C

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 5/20 0.59
ABL1 P00519 1/20 0.58
BCR P11274 1/20 0.58
CYP1A1 P04798 2/20 0.56
PTGS1 P23219 2/20 0.56
PTGS2 P35354 1/20 0.56
LCK P06239 2/20 0.55
APP P05067 4/20 0.54
CYP1A2 P05177 1/20 0.53
CYP1B1 Q16678 1/20 0.53
NQO2 P16083 1/20 0.53
NR1H4 Q96RI1 1/20 0.52
NFE2L2 Q16236 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18648519 1.00 TUBB1 (0.59) TUBB1ABL1BCRCYP1A1PTGS1
SCHEMBL10281431 0.86 PTGS1 (0.74) TUBB1ABL1BCRCYP1A1PTGS1
SCHEMBL15633028 0.85 TUBB1 (0.78) TUBB1ABL1BCRCYP1A1PTGS1
SCHEMBL30609589 0.85 TUBB1 (0.78) TUBB1ABL1BCRCYP1A1PTGS1
SCHEMBL15633027 0.85 TUBB1 (0.78) TUBB1ABL1BCRCYP1A1PTGS1
SCHEMBL14363441 0.84 CYP1A1 (0.73) TUBB1CYP1A1PTGS1PTGS2APP
SCHEMBL20223710 0.83 TUBB1 (0.68) TUBB1CYP1A1PTGS1PTGS2APP
SCHEMBL27305906 0.81 LCK (0.70) TUBB1ABL1BCRPTGS1PTGS2
SCHEMBL5315834 0.79 ABL1 (0.67) TUBB1ABL1BCRCYP1A1PTGS1
SCHEMBL21980865 0.78 TUBB1 (0.71) TUBB1ABL1BCRCYP1A1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-11-03 EP disclosed
WO-2009103626-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed