SCHEMBL3395018

SCHEMBL3395018

COc1cccc(COc2cccc(C=Cc3ccc(OC)c(C)c3)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.58
MAOB P27338 8/20 0.57
LCK P06239 1/20 0.54
MAOA P21397 2/20 0.52
RELA Q04206 1/20 0.51
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50
TUBA1B P68363 1/20 0.50
TUBA4A P68366 1/20 0.50
TUBB4B P68371 1/20 0.50
TUBB3 Q13509 1/20 0.50
TUBB2A Q13885 1/20 0.50
TUBB8 Q3ZCM7 1/20 0.50
TUBA3E Q6PEY2 1/20 0.50
TUBA1A Q71U36 1/20 0.50
TUBA1C Q9BQE3 1/20 0.50
TUBB6 Q9BUF5 1/20 0.50
TUBB2B Q9BVA1 1/20 0.50
TUBB1 Q9H4B7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28586185 0.77 NPC1 (0.78) MAOBMAOANPC1RAB9ATDP1
SCHEMBL2280993 0.76 MRGPRX4 (0.52) MAOBMAOARELANPC1RAB9A
SCHEMBL7534312 0.76 NQO2 (0.58) NQO2RELATUBB4ATUBBTUBA3C
SCHEMBL3394056 0.75 TUBB1 (0.59) NQO2LCKTUBB1NFE2L2CYP1A1
SCHEMBL18648519 0.75 TUBB1 (0.59) NQO2LCKTUBB1NFE2L2CYP1A1
SCHEMBL14989228 0.75 NQO2 (1.00) NQO2RELATUBB4ATUBBTUBA3C
SCHEMBL8264358 0.75 NQO2 (0.74) NQO2TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL13144444 0.73 MAOB (0.87) MAOBMAOA
SCHEMBL14363441 0.73 CYP1A1 (0.73) NQO2TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL16710547 0.73 MAOB (0.71) MAOBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-11-03 EP disclosed
WO-2009103626-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed