SCHEMBL3395528

SCHEMBL3395528

Cc1cc(C#N)ccc1-c1ccnc(NCc2cc(-c3ccc(Br)o3)[nH]n2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.54
IDH1 O75874 2/20 0.34
CLK4 Q9HAZ1 4/20 0.34
CYP1A2 P05177 4/20 0.34
CYP3A4 P08684 4/20 0.34
ALDH1A1 P00352 3/20 0.34
MAPK1 P28482 3/20 0.34
DYRK1A Q13627 1/20 0.33
HSD17B10 Q99714 3/20 0.33
CYP2D6 P10635 2/20 0.33
TSHR P16473 2/20 0.33
CYP2C19 P33261 2/20 0.33
USP2 O75604 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.33
S1PR1 P21453 1/20 0.33
EGLN2 Q96KS0 2/20 0.32
HRH2 P25021 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13425790 0.90 KCNH2 (0.56) KCNH2IDH1CLK4CYP1A2CYP3A4
SCHEMBL13425784 0.86 KCNH2 (0.52) KCNH2IDH1CLK4CYP1A2ALDH1A1
SCHEMBL13425751 0.85 KCNH2 (0.51) KCNH2IDH1CLK4CYP1A2CYP3A4
SCHEMBL13425760 0.85 KCNH2 (0.61) KCNH2IDH1CLK4CYP1A2CYP3A4
SCHEMBL13425792 0.85 KCNH2 (0.61) KCNH2IDH1CLK4CYP1A2CYP3A4
SCHEMBL13425597 0.85 KCNH2 (0.50) KCNH2IDH1CLK4MAPK1DYRK1A
SCHEMBL13425632 0.84 KCNH2 (0.49) KCNH2CLK4MAPK1DYRK1AHRH2
SCHEMBL3432958 0.84 KCNH2 (0.60) KCNH2IDH1CLK4CYP1A2CYP3A4
SCHEMBL13425609 0.83 KCNH2 (0.49) KCNH2CLK4ALDH1A1MAPK1DYRK1A
SCHEMBL13426154 0.83 KCNH2 (0.68) KCNH2CLK4CYP1A2CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed