SCHEMBL3395657

SCHEMBL3395657

CC(=O)[C@@]1(O)CC[C@H]2[C@@H]3C[C@H](C)C4=CC(=O)CC[C@]4(C)[C@H]3[C@@H](O)C[C@@]21C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 10/20 1.00
CYP3A4 P08684 8/20 1.00
HSD17B10 Q99714 4/20 1.00
ALDH1A1 P00352 3/20 1.00
CYP2C9 P11712 2/20 1.00
TSHR P16473 1/20 1.00
NR3C1 P04150 7/20 0.73
LMNA P02545 6/20 0.73
KMT2A Q03164 4/20 0.73
CYP2C19 P33261 3/20 0.73
MAPT P10636 2/20 0.73
MEN1 O00255 2/20 0.73
PGR P06401 6/20 0.65
SMN1; SMN2 Q16637 3/20 0.65
SHBG P04278 2/20 0.56
NR3C2 P08235 2/20 0.56
SERPINA6 P08185 2/20 0.56
NFKB1 P19838 1/20 0.56
AR P10275 3/20 0.55
CHRM1 P11229 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3395660 1.00 HIF1A (1.00) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9
SCHEMBL13069730 1.00 HIF1A (1.00) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9
SCHEMBL17714998 1.00 HIF1A (1.00) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9
SCHEMBL8637937 1.00 HIF1A (1.00) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9
SCHEMBL3406165 0.92 HIF1A (0.85) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9
SCHEMBL137529 0.89 KMT2A (0.84) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9
SCHEMBL17714999 0.89 KMT2A (0.84) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9
SCHEMBL13150977 0.89 KMT2A (0.84) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9
SCHEMBL137530 0.89 KMT2A (0.84) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9
SCHEMBL10393880 0.89 KMT2A (0.84) HIF1ACYP3A4HSD17B10ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4041055-A SULFENYLATION, MICHAEL ADDITION, REACTION WITH THIOPHILE, HYDROLYSIS THE UPJOHN COMPANY (US) 1977-08-09 US claimed
CN-116410939-A 3-sterone-delta 1 Dehydrogenase mutant and application thereof in synthesis of steroid C1,2 dehydrogenation drug intermediates 中国科学院天津工业生物技术研究所 2023-07-11 CN disclosed
EP-2246359-A1 Process for obtaining fluorometholone and intermediates therefor Crystal Pharma, S.L.U. (ES) 2010-11-03 EP disclosed