SCHEMBL3395884

SCHEMBL3395884

Oc1ccc(C=Cc2cccc(Br)c2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.71
APP P05067 3/20 0.61
NPC1 O15118 2/20 0.56
MTOR P42345 2/20 0.56
HSD17B3 P37058 1/20 0.56
TTR P02766 2/20 0.56
TRPA1 O75762 2/20 0.55
MAOB P27338 3/20 0.54
MAOA P21397 2/20 0.54
NQO2 P16083 2/20 0.53
LCK P06239 1/20 0.53
ALDH1A1 P00352 3/20 0.52
CA12 O43570 2/20 0.52
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
CA3 P07451 2/20 0.52
CA4 P22748 2/20 0.52
CA6 P23280 2/20 0.52
CA5A P35218 2/20 0.52
CA7 P43166 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27557619 0.86 LCK (0.67) BACE1NPC1HSD17B3MAOBLCK
SCHEMBL699611 0.85 HSD17B3 (0.57) BACE1HSD17B3MAOBMAOAALDH1A1
SCHEMBL699610 0.85 HSD17B3 (0.57) BACE1HSD17B3MAOBMAOAALDH1A1
SCHEMBL8900696 0.85 HSD17B3 (0.57) BACE1HSD17B3MAOBMAOAALDH1A1
SCHEMBL1931278 0.85 APP (0.73) APPNPC1MTORTTRTRPA1
SCHEMBL8900441 0.85 HSD17B3 (0.65) BACE1HSD17B3MAOBMAOAALDH1A1
SCHEMBL699462 0.85 HSD17B3 (0.65) BACE1HSD17B3MAOBMAOAALDH1A1
SCHEMBL709614 0.85 HSD17B3 (0.65) BACE1HSD17B3MAOBMAOAALDH1A1
SCHEMBL3219281 0.84 BACE1 (1.00) BACE1HSD17B3MAOBMAOAABCB1
SCHEMBL3219293 0.84 BACE1 (1.00) BACE1HSD17B3MAOBMAOAABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-11-03 EP disclosed
WO-2009103626-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed