SCHEMBL3396366

SCHEMBL3396366

COC(=O)c1cccc(NC(=O)C2CCCN(Cc3ccccc3)C2)c1O

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 5/20 0.56
KDM4E B2RXH2 6/20 0.55
ALDH1A1 P00352 3/20 0.55
SCN4A P35499 2/20 0.53
HPGD P15428 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
LMNA P02545 2/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
TSHR P16473 1/20 0.50
BCHE P06276 1/20 0.49
ACHE P22303 1/20 0.49
MAOB P27338 1/20 0.49
DRD4 P21917 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401190 0.90 MEN1 (0.54) HSD17B10KDM4EALDH1A1SCN4AHPGD
SCHEMBL3401687 0.88 KDM4E (0.61) HSD17B10KDM4EALDH1A1SCN4AHPGD
SCHEMBL206309 0.83 HSD17B10 (0.55) HSD17B10KDM4EALDH1A1HPGDNPSR1
SCHEMBL3434303 0.82 NPSR1 (0.66) HSD17B10KDM4EALDH1A1HPGDNPSR1
SCHEMBL5121387 0.77 KDM4E (0.67) HSD17B10KDM4EKMT2AMEN1GAA
SCHEMBL206204 0.77 SMN1; SMN2 (0.62) HSD17B10KDM4EALDH1A1HPGDNPSR1
SCHEMBL206214 0.76 KDM4E (0.49) HSD17B10KDM4EALDH1A1HPGDNPSR1
SCHEMBL29333202 0.76 KDM4E (0.67) KDM4EALDH1A1HPGDKMT2AMEN1
SCHEMBL21653205 0.75 SCN4A (0.57) KDM4EALDH1A1SCN4AHPGDKMT2A
SCHEMBL206203 0.75 KDM4E (0.46) HSD17B10KDM4EALDH1A1HPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247600-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) Lead Therapeutics, Inc. (US) 2010-11-10 EP disclosed
WO-2009099736-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) LEAD THERAPEUTICS, INC. (US) 2009-08-13 WO disclosed