SCHEMBL3396582

SCHEMBL3396582

Clc1ccc2c(n1)[nH]c1ccc(C#CC3CCCCC3)cc12.Clc1ccc2c(n1)[nH]c1ccc(C#Cc3ccccc3)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIKFYVE Q9Y2I7 2/20 0.38
HAO1 Q9UJM8 3/20 0.35
MAPT P10636 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
PTGES O14684 3/20 0.35
CYP1A2 P05177 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GMNN O75496 1/20 0.35
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
TSHR P16473 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
CYP2C19 P33261 1/20 0.35
MTOR P42345 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
HIF1A Q16665 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL674727 0.94 PIKFYVE (0.41) PIKFYVEHAO1MAPTNPC1RAB9A
SCHEMBL676917 0.87 KDM4E (0.44) MAPTCYP1A2KDM4EGMNNLMNA
SCHEMBL676121 0.76 PIKFYVE (0.43) PIKFYVEMAPTNPC1RAB9ACYP1A2
SCHEMBL675083 0.73 ALK (0.45) PIKFYVEMAPTNPC1RAB9ACYP1A2
SCHEMBL675871 0.72 NPC1 (0.43) PIKFYVEMAPTNPC1RAB9ACYP1A2
SCHEMBL11225320 0.69 CYP1A2 (0.55) HAO1MAPTNPC1RAB9APTGES
SCHEMBL8752132 0.69 CYP1A2 (0.55) HAO1MAPTNPC1RAB9APTGES
SCHEMBL676829 0.69 CHRNB2 (0.36) PIKFYVEHAO1MAPTNPC1RAB9A
SCHEMBL675919 0.68 KDM4E (0.54) NPC1PTGESCYP1A2KDM4EGMNN
SCHEMBL11232546 0.68 FFAR1 (0.53) HAO1MAPTNPC1RAB9APTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025872-A2 ALFA-CARBOLINE INHIBITORS OF NPM-ALK, RET, AND BCR-ABL UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2010-03-11 WO disclosed