SCHEMBL3398545

SCHEMBL3398545

CS(=O)(=O)c1ccc(-c2nc(C(F)(F)F)nc(N3CCOCC3)c2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.58
PDE4B Q07343 1/20 0.58
PDE4C Q08493 1/20 0.58
PDE4D Q08499 1/20 0.58
SLC2A1 P11166 1/20 0.46
MTOR P42345 4/20 0.44
PIK3CA P42336 1/20 0.43
PIK3CG P48736 1/20 0.43
GHSR Q92847 1/20 0.43
PTGS2 P35354 8/20 0.43
PTGS1 P23219 5/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2085106 0.88 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DMTOR
SCHEMBL2086343 0.88 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DPTGS2
SCHEMBL14852792 0.81 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DPTGS2
SCHEMBL2085527 0.81 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DMTOR
SCHEMBL1573242 0.80 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL14852793 0.79 BCL2 (0.47) PDE4APDE4BPDE4CPDE4DPTGS2
SCHEMBL17970604 0.79 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DPTGS2
SCHEMBL12936298 0.79 PTGS2 (0.47) PDE4APDE4BPDE4CPDE4DPTGS2
SCHEMBL2083337 0.79 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DPTGS2
SCHEMBL12936302 0.78 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8420653-B2 Pyrimidine compounds and their uses ORCHID CHEMICALS & PHARMACEUTICALS LIMITED (IN) 2013-04-16 US claimed
EP-2245017-A2 NOVEL HETEROCYCLES Orchid Research Laboratories Limited (IN) 2010-11-03 EP disclosed
WO-2009095773-A2 NOVEL HETEROCYCLES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2009-08-06 WO disclosed