SCHEMBL3398671

SCHEMBL3398671

Cc1nc(-c2ccc(N(C)C)cc2)sc1C(=O)NCCC1CCCN1C

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.53
CHRM4 P08173 4/20 0.52
CHRM3 P20309 1/20 0.47
NPC1 O15118 1/20 0.44
HPGD P15428 1/20 0.44
PPARA Q07869 6/20 0.43
GAA P10253 2/20 0.42
PPARD Q03181 4/20 0.42
PPARG P37231 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3399976 0.89 ACKR3 (0.52) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3405398 0.89 ACKR3 (0.55) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3401785 0.88 ACKR3 (0.54) ACKR3CHRM4CHRM3NPC1HPGD
SCHEMBL3399830 0.88 ACKR3 (0.54) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3403598 0.87 ACKR3 (0.53) ACKR3CHRM4CHRM3PPARAPPARD
SCHEMBL3405823 0.87 ACKR3 (0.53) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3403460 0.87 CHRM4 (0.54) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3403946 0.87 CHRM4 (0.56) ACKR3CHRM4CHRM3NPC1HPGD
SCHEMBL3405198 0.86 CHRM4 (0.67) ACKR3CHRM4CHRM3NPC1PPARA
SCHEMBL3405442 0.86 ACKR3 (0.59) ACKR3CHRM4NPC1HPGDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed