SCHEMBL3399147

SCHEMBL3399147

COc1ccc(-c2cc(CNc3cc(-c4ccc(C#N)cc4C)ccn3)n[nH]2)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.56
CLK4 Q9HAZ1 4/20 0.40
DYRK1A Q13627 1/20 0.40
CHEK1 O14757 2/20 0.38
USP2 O75604 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
TSHR P16473 2/20 0.38
CYP2C19 P33261 2/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
GLA P06280 1/20 0.38
CYP2C9 P11712 1/20 0.38
PDE5A O76074 3/20 0.38
IDH1 O75874 1/20 0.37
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13426232 0.90 KCNH2 (0.55) KCNH2CLK4DYRK1ACHEK1USP2
SCHEMBL13426222 0.89 KCNH2 (0.59) KCNH2CLK4DYRK1AUSP2ALDH1A1
SCHEMBL13425582 0.89 KCNH2 (0.56) KCNH2CLK4DYRK1ACHEK1USP2
SCHEMBL13426219 0.89 KCNH2 (0.58) KCNH2CLK4DYRK1AALDH1A1CYP1A2
SCHEMBL3398430 0.88 KCNH2 (0.58) KCNH2CLK4DYRK1ACHEK1USP2
SCHEMBL13426255 0.88 KCNH2 (0.57) KCNH2CLK4DYRK1ACHEK1USP2
SCHEMBL13425826 0.88 KCNH2 (0.64) KCNH2CLK4DYRK1ACHEK1USP2
SCHEMBL3397557 0.87 KCNH2 (0.59) KCNH2CLK4DYRK1AUSP2ALDH1A1
SCHEMBL13425837 0.86 KCNH2 (0.54) KCNH2CLK4DYRK1ACHEK1USP2
SCHEMBL3397173 0.85 KCNH2 (0.58) KCNH2CLK4DYRK1ACHEK1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed