SCHEMBL3399266

SCHEMBL3399266

C=C(c1cccc(C)c1)c1cccc(Br)c1.Cc1cccc(C2(c3cccc(Br)c3)COC(N)=N2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 11/20 0.39
CTSD P07339 6/20 0.39
TAAR1 Q96RJ0 1/20 0.38
CHRNA1 P02708 2/20 0.36
CHRNG P07510 2/20 0.36
CHRNB1 P11230 2/20 0.36
CHRNB2 P17787 2/20 0.36
SLC6A2 P23975 2/20 0.36
CHRNB4 P30926 2/20 0.36
CHRNA3 P32297 2/20 0.36
CHRNA4 P43681 2/20 0.36
SLC6A3 Q01959 2/20 0.36
CHRND Q07001 2/20 0.36
CTSL P07711 1/20 0.36
SLC6A4 P31645 1/20 0.36
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2276540 0.89 BACE1 (0.46) BACE1CTSDTAAR1CHRNA1CHRNG
SCHEMBL2276542 0.89 BACE1 (0.46) BACE1CTSDTAAR1CHRNA1CHRNG
SCHEMBL3398703 0.83 BACE1 (0.41) BACE1CTSDTAAR1CTSLMEN1
SCHEMBL3398692 0.81 BACE1 (0.46) BACE1CTSDTAAR1
SCHEMBL3393923 0.80 BACE1 (0.47) BACE1CTSDTAAR1MEN1GAA
SCHEMBL3393576 0.79 BACE1 (0.44) BACE1CTSDTAAR1
SCHEMBL3399127 0.79 BACE1 (0.54) BACE1CTSDTAAR1
SCHEMBL2285631 0.78 BACE1 (0.49) BACE1CTSDTAAR1
SCHEMBL2285635 0.78 BACE1 (0.49) BACE1CTSDTAAR1
SCHEMBL3399227 0.77 BACE1 (0.36) BACE1CTSDTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-11-03 EP disclosed
WO-2009103626-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed