SCHEMBL3399284

SCHEMBL3399284

CS(=O)(=O)c1ccc(-c2ccnc(C(F)(F)F)n2)cc1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.52
KCNH2 Q12809 2/20 0.49
PTGS1 P23219 7/20 0.48
SYK P43405 1/20 0.45
MAP4K4 O95819 1/20 0.45
PIK3CA P42336 1/20 0.45
MINK1 Q8N4C8 1/20 0.45
PI4KB Q9UBF8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28175534 0.80 PIK3CA (0.44) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL16826895 0.76 PTGS2 (0.56) PTGS2KCNH2
SCHEMBL3754393 0.76 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL3157555 0.76 PTGS2 (0.52) PTGS2KCNH2PTGS1
SCHEMBL27999249 0.76 AAK1 (0.44) SYK
SCHEMBL28886728 0.75 AURKA (0.53)
SCHEMBL31475459 0.74 MALT1 (0.40) PTGS2KCNH2SYKMAP4K4PIK3CA
SCHEMBL16538788 0.74 KCNH2 (0.53) PTGS2KCNH2PTGS1SYKMAP4K4
SCHEMBL22340390 0.73 IDH1 (0.35)
SCHEMBL18963 0.73 NPSR1 (0.49) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245017-A2 NOVEL HETEROCYCLES Orchid Research Laboratories Limited (IN) 2010-11-03 EP claimed
WO-2009095773-A2 NOVEL HETEROCYCLES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2009-08-06 WO claimed
EP-1973884-A2 NOVEL HETEROCYCLES Orchid Research Laboratories Limited (IN) 2008-10-01 EP claimed
WO-2007083182-A2 NOVEL HETEROCYCLES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-07-26 WO claimed