SCHEMBL3399343

SCHEMBL3399343

COc1cc(F)ccc1C(=O)NC1COCCn2c1nc(-c1ccncn1)cc2=O

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 0.47
CYP2D6 P10635 8/20 0.47
CYP1A2 P05177 5/20 0.47
CSNK1A1 P48729 1/20 0.39
GSK3A P49840 1/20 0.39
MTOR P42345 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402193 0.92 GSK3B (0.42) GSK3BCYP2D6CYP1A2MTOR
SCHEMBL3402173 0.91 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL927355 0.91 GSK3B (0.39) GSK3BCYP2D6CYP1A2MTOR
SCHEMBL3399684 0.91 CRBN (0.42) GSK3BCYP2D6CYP1A2MTOR
SCHEMBL2065707 0.90 GSK3B (0.50) GSK3BCYP2D6CYP1A2
SCHEMBL3397799 0.90 GSK3B (0.44) GSK3BCYP2D6CYP1A2MTOR
SCHEMBL2064913 0.89 GSK3B (0.49) GSK3BCYP2D6CYP1A2
SCHEMBL2065317 0.88 GSK3B (0.48) GSK3BCYP2D6CYP1A2
SCHEMBL3399573 0.88 GSK3B (0.44) GSK3BCYP2D6CYP1A2
SCHEMBL3400870 0.87 GSK3B (0.42) GSK3BCYP2D6CYP1A2MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247599-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP claimed
WO-2009095788-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO claimed
EP-2247599-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP disclosed
WO-2009095788-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO disclosed