SCHEMBL3400870

SCHEMBL3400870

COc1ccc(OC)c(C(=O)NC2COCCn3c2nc(-c2ccncn2)cc3=O)c1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 17/20 0.42
CYP2D6 P10635 6/20 0.42
CYP1A2 P05177 5/20 0.40
CYP3A4 P08684 3/20 0.40
MTOR P42345 1/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402193 0.94 GSK3B (0.42) GSK3BCYP2D6CYP1A2CYP3A4MTOR
SCHEMBL3425658 0.92 KCNMA1 (0.40) GSK3BCYP2D6CYP1A2MTOR
SCHEMBL3402010 0.92 GSK3B (0.39) GSK3BCYP2D6CYP1A2CYP3A4MTOR
SCHEMBL3402173 0.91 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL3402360 0.89 POLB (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL2064445 0.88 GSK3B (0.41) GSK3BCYP2D6CYP1A2CYP3A4HCRTR1
SCHEMBL3399343 0.87 GSK3B (0.47) GSK3BCYP2D6CYP1A2MTOR
SCHEMBL3399573 0.87 GSK3B (0.44) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL927355 0.87 GSK3B (0.39) GSK3BCYP2D6CYP1A2MTOR
SCHEMBL3399684 0.87 CRBN (0.42) GSK3BCYP2D6CYP1A2CYP3A4MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247599-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP claimed
WO-2009095788-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO claimed
EP-2247599-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP disclosed
WO-2009095788-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO disclosed