SCHEMBL3399377

SCHEMBL3399377

CN(C)CCCOc1ccc(-c2ccc3[nH]c4ncc(Cl)cc4c3c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.47
CXCR1 P25024 2/20 0.46
ACHE P22303 3/20 0.45
MAOA P21397 1/20 0.43
ATM Q13315 2/20 0.42
CHEK2 O96017 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TLR9 Q9NR96 1/20 0.41
TLR8 Q9NR97 1/20 0.41
TLR7 Q9NYK1 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
ALOX5 P09917 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
ATR Q13535 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL675132 0.89 ACHE (0.47) ACHESMN1; SMN2KDM4ENPC1RAB9A
SCHEMBL675184 0.83 LSS (0.46) LSSCXCR1ACHEMAOAATM
SCHEMBL3733141 0.83 LSS (0.42) LSSMAOAATMCHEK2SMN1; SMN2
SCHEMBL676066 0.81 ALK (0.53) LSSCXCR1ACHEMAOAATM
SCHEMBL675220 0.81 ALK (0.48) ACHEKDM4EALDH1A1HSD17B10
SCHEMBL3725897 0.80 LSS (0.39) LSSMAOAATMCHEK2SMN1; SMN2
SCHEMBL3725895 0.80 LSS (0.39) LSSMAOAATMCHEK2SMN1; SMN2
SCHEMBL6220994 0.79 LSS (0.52) LSSCXCR1ACHE
SCHEMBL6503218 0.79 TNK2 (0.47) LSSCXCR1ACHEMAOACHEK2
SCHEMBL675056 0.79 HRH4 (0.52) CXCR1ACHETLR8TLR7NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025872-A2 ALFA-CARBOLINE INHIBITORS OF NPM-ALK, RET, AND BCR-ABL UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2010-03-11 WO disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed