SCHEMBL3399483

SCHEMBL3399483

CCc1cccc(CC)c1-c1nc(C)c(CN2CCN(C(C)C)CC2)s1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
GNRHR P30968 1/20 0.35
GPR4 P46093 4/20 0.34
HRH3 Q9Y5N1 7/20 0.34
KCNH2 Q12809 3/20 0.34
TACR2 P21452 2/20 0.34
TACR3 P29371 1/20 0.34
MAOB P27338 2/20 0.33
HCN4 Q9Y3Q4 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
KDM1A O60341 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400874 0.96 HRH3 (0.36) KDM4EALDH1A1TDP1BCHEACHE
SCHEMBL13072167 0.89 KMT2A (0.39) KDM4EGNRHR
SCHEMBL3404520 0.81 TACR2 (0.43) KDM4EHRH3KCNH2TACR2TACR3
SCHEMBL3400819 0.78 HTR2C (0.46) KDM4EALDH1A1MAOB
SCHEMBL3405240 0.75 HTR2C (0.45) KDM4EALDH1A1TACR2
SCHEMBL5929244 0.73 RXFP1 (0.40) KDM4EALDH1A1KCNH2
SCHEMBL12030410 0.67 TACR2 (0.46) KDM4EALDH1A1HRH3KCNH2TACR2
SCHEMBL18705076 0.67 CXCR4 (0.46) KDM4EALDH1A1TDP1BCHEACHE
SCHEMBL5928960 0.67 GABRA1 (0.42) KDM4EALDH1A1KCNH2
Hydrochloric Acid SCHEMBL2484779 0.67 TACR2 (0.45) KDM4EALDH1A1HRH3KCNH2TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed