SCHEMBL3399574

SCHEMBL3399574

CN1CCCN(c2cccc(Cl)c2Cl)CC1

nearest known ligand 0.87

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 15/20 0.87
DRD3 P35462 14/20 0.87
DRD4 P21917 5/20 0.58
HTR1A P08908 2/20 0.58
HTR2A P28223 1/20 0.58
HTR2C P28335 1/20 0.58
BCL2A1 Q16548 1/20 0.56
ADRB1 P08588 1/20 0.56
NCF1 P14598 1/20 0.53
LMNA P02545 1/20 0.51
KMT2A Q03164 1/20 0.51
DRD5 P21918 1/20 0.50
ADRA2C P18825 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3399254 0.93 DRD2 (1.00) DRD2DRD3DRD4HTR1AHTR2A
SCHEMBL8452211 0.84 DRD2 (0.69) DRD2DRD3DRD4ADRB1DRD5
SCHEMBL2131518 0.82 DRD2 (0.67) DRD2DRD3DRD4ADRB1DRD5
SCHEMBL30751119 0.82 DRD2 (0.67) DRD2DRD3DRD4ADRB1DRD5
SCHEMBL3395428 0.81 DRD2 (0.62) DRD2DRD3DRD4HTR1AADRB1
SCHEMBL21599144 0.81 DRD2 (0.56) DRD2DRD3DRD4HTR1AHTR2A
SCHEMBL24399496 0.80 KDM4E (0.75) DRD2DRD3DRD4HTR1AHTR2A
SCHEMBL22302770 0.80 DRD2 (0.89) DRD2DRD3DRD4HTR1AHTR2A
SCHEMBL424507 0.80 DRD2 (0.75) DRD2DRD3DRD4HTR1AHTR2A
SCHEMBL12359055 0.77 DRD2 (0.71) DRD2DRD3DRD4HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003418-A2 FUNCTIONALLY SELECTIVE LIGANDS OF DOPAMINE D2 RECEPTORS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2012-01-05 WO disclosed