SCHEMBL3399982

SCHEMBL3399982

Cc1nc(-c2ccc(OC(F)(F)F)cc2)sc1C(=O)NCCC1CCCN1C

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 12/20 0.57
PPARD Q03181 5/20 0.57
CHRM4 P08173 4/20 0.54
ACKR3 P25106 1/20 0.51
PPARG P37231 2/20 0.49
CHRM3 P20309 1/20 0.49
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401785 0.91 ACKR3 (0.54) PPARAPPARDCHRM4ACKR3PPARG
SCHEMBL3398440 0.91 ACKR3 (0.51) PPARAPPARDCHRM4ACKR3CHRM3
SCHEMBL3403598 0.90 ACKR3 (0.53) PPARAPPARDCHRM4ACKR3PPARG
SCHEMBL3405442 0.89 ACKR3 (0.59) PPARAPPARDCHRM4ACKR3NPC1
SCHEMBL3405198 0.89 CHRM4 (0.67) PPARAPPARDCHRM4ACKR3PPARG
SCHEMBL3405220 0.88 ACKR3 (0.52) PPARAPPARDCHRM4ACKR3NPC1
SCHEMBL3405398 0.88 ACKR3 (0.55) PPARAPPARDCHRM4ACKR3PPARG
SCHEMBL13310379 0.87 ACKR3 (0.50) PPARAPPARDCHRM4ACKR3PPARG
SCHEMBL3403946 0.86 CHRM4 (0.56) PPARAPPARDCHRM4ACKR3PPARG
SCHEMBL3402589 0.86 ACKR3 (0.51) PPARAPPARDCHRM4ACKR3PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed