SCHEMBL3400299

SCHEMBL3400299

COC(=O)c1cccc(N(C(=O)OCc2ccccc2)C(=O)C2CCNCC2)c1OC(=O)C1CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
HTT P42858 1/20 0.44
CYP2C19 P33261 1/20 0.43
GRIN2B Q13224 7/20 0.39
ENPP2 Q13822 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400302 0.77 SMN1; SMN2 (0.58) SMN1; SMN2NPC1RAB9AHTTCYP2C19
SCHEMBL26925420 0.71 SMN1; SMN2 (0.71) SMN1; SMN2NPC1RAB9AHTTCYP2C19
SCHEMBL485156 0.71 SMN1; SMN2 (0.75) SMN1; SMN2NPC1RAB9AHTTCYP2C19
SCHEMBL12699823 0.71 SMN1; SMN2 (0.67) SMN1; SMN2NPC1RAB9AHTTCYP2C19
SCHEMBL206538 0.69 SMN1; SMN2 (0.59) SMN1; SMN2NPC1RAB9AHTTCYP2C19
SCHEMBL351651 0.68 SMN1; SMN2 (0.73) SMN1; SMN2NPC1RAB9AHTTCYP2C19
SCHEMBL30711214 0.68 SMN1; SMN2 (0.60) SMN1; SMN2NPC1RAB9AHTTCYP2C19
SCHEMBL895470 0.68 SMN1; SMN2 (0.68) SMN1; SMN2NPC1RAB9AHTTCYP2C19
SCHEMBL31170142 0.68 SMN1; SMN2 (0.69) SMN1; SMN2NPC1RAB9AHTTCYP2C19
SCHEMBL31170255 0.68 SMN1; SMN2 (0.69) SMN1; SMN2NPC1RAB9AHTTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247600-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) Lead Therapeutics, Inc. (US) 2010-11-10 EP disclosed
WO-2009099736-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) LEAD THERAPEUTICS, INC. (US) 2009-08-13 WO disclosed