SCHEMBL3400302

SCHEMBL3400302

COC(=O)c1cccc(NC(=O)C2CCN(C(=O)OCc3ccccc3)CC2)c1OC(=O)C1CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.58
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
HTT P42858 1/20 0.56
ENPP2 Q13822 3/20 0.52
HSD17B10 Q99714 5/20 0.51
KDM4E B2RXH2 4/20 0.51
CYP2C19 P33261 2/20 0.51
TSHR P16473 2/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
MAPK1 P28482 1/20 0.51
MAPT P10636 1/20 0.50
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
POLB P06746 2/20 0.47
ACHE P22303 1/20 0.43
BACE1 P56817 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206204 0.87 SMN1; SMN2 (0.62) SMN1; SMN2NPC1RAB9AHTTENPP2
SCHEMBL205824 0.82 SMN1; SMN2 (0.56) SMN1; SMN2NPC1RAB9AHTTENPP2
SCHEMBL28268704 0.78 SMN1; SMN2 (0.61) SMN1; SMN2NPC1RAB9AHTTENPP2
SCHEMBL206309 0.78 HSD17B10 (0.55) SMN1; SMN2NPC1RAB9AHTTHSD17B10
SCHEMBL485156 0.78 SMN1; SMN2 (0.75) SMN1; SMN2NPC1RAB9AHTTENPP2
SCHEMBL2306241 0.77 SMN1; SMN2 (0.68) SMN1; SMN2NPC1RAB9AHTTENPP2
SCHEMBL206214 0.77 KDM4E (0.49) SMN1; SMN2NPC1RAB9AHTTHSD17B10
SCHEMBL12699823 0.77 SMN1; SMN2 (0.67) SMN1; SMN2NPC1RAB9AHTTENPP2
SCHEMBL3400299 0.77 SMN1; SMN2 (0.46) SMN1; SMN2NPC1RAB9AHTTENPP2
SCHEMBL5272899 0.77 KDM4E (0.60) SMN1; SMN2NPC1RAB9AHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247600-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) Lead Therapeutics, Inc. (US) 2010-11-10 EP disclosed
WO-2009099736-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) LEAD THERAPEUTICS, INC. (US) 2009-08-13 WO disclosed