SCHEMBL3400558

SCHEMBL3400558

NC(=O)c1cccc2nc(C3CCN(Cc4ccccc4)CC3)oc12

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.47
PARP1 P09874 5/20 0.46
USP2 O75604 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ACHE P22303 2/20 0.45
GAA P10253 1/20 0.45
OPRK1 P41145 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
BCHE P06276 1/20 0.43
DRD2 P14416 1/20 0.43
HTR6 P50406 1/20 0.43
PARP2 Q9UGN5 2/20 0.42
PARP3 Q9Y6F1 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL203957 0.84 PARP1 (0.57) PARP1LMNADRD2PARP2
SCHEMBL206528 0.83 SMN1; SMN2 (0.53) USP2ALDH1A1TSHRNPSR1LMNA
SCHEMBL207485 0.82 PARP1 (0.50) PARP1LMNAPARP2
SCHEMBL205714 0.81 PARP1 (0.49) DRD4PARP1LMNADRD2PARP2
SCHEMBL204714 0.77 PARP1 (0.51) PARP1ALDH1A1PARP2
SCHEMBL27969428 0.77 BCHE (0.59) DRD4USP2ALDH1A1TSHRNPSR1
SCHEMBL206737 0.77 LCK (0.46) NPSR1
SCHEMBL5621740 0.77 HTR2B (0.54) DRD4PARP1ALDH1A1GAAPARP2
SCHEMBL205895 0.76 SMN1; SMN2 (0.44) PARP1NPSR1PARP2
SCHEMBL14157392 0.76 CHRM4 (0.46) DRD4USP2ALDH1A1TSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247600-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) Lead Therapeutics, Inc. (US) 2010-11-10 EP disclosed
WO-2009099736-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) LEAD THERAPEUTICS, INC. (US) 2009-08-13 WO disclosed