SCHEMBL3400734

SCHEMBL3400734

CS(=O)(=O)CCn1ccc2ncnc(Cl)c21

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 2/20 0.39
FGFR4 P22455 1/20 0.39
EGFR P00533 12/20 0.36
ERBB2 P04626 12/20 0.36
KDR P35968 6/20 0.34
ERBB3 P21860 3/20 0.34
ERBB4 Q15303 3/20 0.34
LPAR1 Q92633 1/20 0.32
LPAR2 Q9HBW0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2749135 0.80 FGFR1 (0.40) FGFR1FGFR4EGFRERBB2KDR
SCHEMBL2749873 0.79 EGFR (0.56) FGFR1FGFR4EGFRERBB2ERBB3
SCHEMBL3403862 0.79 FGFR1 (0.40) FGFR1FGFR4EGFRERBB2KDR
SCHEMBL3506358 0.78 FGFR1 (0.39) FGFR1FGFR4EGFRERBB2KDR
SCHEMBL2748776 0.77 FGFR1 (0.40) FGFR1FGFR4EGFRERBB2ERBB3
SCHEMBL2749352 0.77 EGFR (0.44) FGFR1FGFR4EGFRERBB2KDR
SCHEMBL2748523 0.77 FGFR1 (0.42) FGFR1FGFR4EGFRERBB2KDR
SCHEMBL27684259 0.77 FGFR1 (0.42) FGFR1FGFR4EGFRERBB2ERBB3
SCHEMBL2747761 0.77 FGFR1 (0.41) FGFR1FGFR4KDR
SCHEMBL3829641 0.77 FGFR1 (0.44) FGFR1FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2253633-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2010-11-24 EP disclosed
US-20090233937-A1 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233937-A1 FUSED HETEROCYCLIC COMPOUND ROS1, JAK2, ERBB2 FGFR1 9/4885FGFR4 54/4885EGFR 11/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.